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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T5829 | H4 Receptor antagonist 1 | Histamine Receptor | |
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. | |||
T38634 | Histamine H4 receptor antagonist-1 | Histamine H4 receptor antagonist-1 | |
Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor. | |||
T11532 | H4R antagonist 1 | Histamine Receptor | |
H4R antagonist 1 is a highly selective histamine H4 receptor (H4R) antagonist (IC50: 27 nM). H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R. | |||
T79786 | H4R antagonist 2 | Histamine Receptor | |
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and holds potential for research into rheumatoid arthritis [1] (page 68). | |||
T61011 | Izuforant | ||
Izuforant (JW1601) (Compound 24) has potent anti-inflammatory and anti-pruritic activities. Izuforant has a binding affinity for human serotonin 3 receptor (h5-HT3R) with an IC50 value of 9.1 μM. Izuforant is also an ora... | |||
T38323 | A-943931 (hydrochloride hydrate) | ||
A-943931 is a histamine H4receptor antagonist (Ki= 3.8 nM).1In vivo, A-943931 inhibits scratching induced by clobenpropit in mice (ED50= 26 μmoles/kg, i.p.). 1.Milicic, I., Witte, D.G., Miller, T.L., et al.Identification... |